Meclinertant

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Meclinertant
SR-48692 structure.png
Systematic (IUPAC) name
2-([1-(7-Chloro-4-quinolinyl)-5-(2,6-dimethoxyphenyl)-1H-pyrazole-3-carbonyl]amino)admantane-2-carboxylic acid
Identifiers
CAS Number 146362-70-1 YesY
PubChem CID: 119192
IUPHAR/BPS 1582
UNII 5JBP4SI96H YesY
ChEMBL CHEMBL506981
Chemical data
Formula C32H31ClN4O5
Molecular mass 587.064
  • c7cc3c(cc7Cl)nccc3-n4nc(cc4-c1c(OC)cccc1OC)C(=O)NC2(C(O)=O)C5CC(C6)CC2CC6C5
  (verify)

Meclinertant (SR-48692) is a drug which acts as a selective, non-peptide antagonist at the neurotensin receptor NTS1, and was the first non-peptide antagonist developed for this receptor.[1][2] It is used in scientific research to explore the interaction between neurotensin and other neurotransmitters in the brain,[3][4][5][6][7][8] and produces anxiolytic, anti-addictive and memory-impairing effects in animal studies.[9][10][11][12]

References

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  1. REDIRECT Template:Peptide receptor modulators


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